| 78件の論文が見つかりました。論文は出版年月日順に表示しています。(ヘルプ) | |
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| Shiho Tsutsumi, Yuki Takechi-Haraya, Yasuhiro Abe, Kohsaku Kawakami. Impact of Lipid Bilayer Composition and Physicochemical Properties on Constitution of a Transmembrane Helical Peptide into Exosome-Mimetic Vesicles. Molecular Pharmaceutics. 22 [11] (2025) 6874-6886 10.1021/acs.molpharmaceut.5c00825 Open Access | |
| Katsutoshi Yamaguchi, Yuya Ishizuka, Etsushi Yoshikawa, Takashi Makishima, Ryo Mizoguchi, Kohsaku Kawakami. Nucleation in Amorphous Terfenadine at a Temperature Much Lower than the Glass Transition Temperature and Its Impact on Physical Stability. Molecular Pharmaceutics. 22 [10] (2025) 6038-6049 10.1021/acs.molpharmaceut.5c00700 Open Access | |
| Toru Yoshitomi, Kyoko Hayashi, Tamasa Araki, Takeshi Annoura, Yukio Nagasaki. Self-Assembling Antioxidant Nanoparticles Increase Survival and Reduce Disease Symptoms of Severe Malaria. Molecular Pharmaceutics. 22 [10] (2025) 5879-5886 10.1021/acs.molpharmaceut.5c00419 | |
| Tianjiao Zeng, Chengyu Lu, Man Wang, Huajian Chen, Toru Yoshitomi, Naoki Kawazoe, Yingnan Yang, Guoping Chen. Long-term exposure in high viscous microenvironment facilitates acquired drug resistance of colon cancer cells to doxorubicin. European Journal of Pharmaceutics and Biopharmaceutics. 216 (2025) 114852 10.1016/j.ejpb.2025.114852 | |
| Dani Lakshman Yarlagadda, Kohsaku Kawakami, Satyavrata Samavedi. Leveraging Molecular Interactions to Develop a Generalized Design Framework for Coamorphous Drug–Drug Mixtures Exhibiting Elevated Glass Transition Temperatures. Molecular Pharmaceutics. 22 [6] (2025) 3084-3096 10.1021/acs.molpharmaceut.5c00006 | |
| Xue Han, Kohsaku Kawakami. Influence of Pore Size of Mesoporous Silica on Physical Stability of Overloaded Celecoxib Glass. Molecular Pharmaceutics. 22 [5] (2025) 2556-2567 10.1021/acs.molpharmaceut.4c01482 Open Access | |
| Kohsaku Kawakami. Roles of Supersaturation and Liquid–Liquid Phase Separation for Enhanced Oral Absorption of Poorly Soluble Drugs from Amorphous Solid Dispersions. Pharmaceutics. 17 [2] (2025) 262 10.3390/pharmaceutics17020262 Open Access | |
| Michinori Oikawa, Satoru Matsuura, Takeyuki Okudaira, Ryo Ito, Kanako Arima, Masahiro Fushimi, Takamasa Oda, Kaoru Ohyama, Kohsaku Kawakami. Bridging the gap between in vitro and in vivo solubility-permeability interplay. Journal of Pharmaceutical Sciences. 114 [1] (2025) 361-370 10.1016/j.xphs.2024.10.008 Open Access | |
| Kohsaku Kawakami, Taichi Ishitsuka, Masafumi Fukiage, Yohei Nishida, Tetsuo Shirai, Yosuke Hirai, Tetsu Hideshima, Fumiaki Tanabe, Koji Shinoda, Ryota Tamate, Takuya Fujita. Long-term physical stability of amorphous solid dispersions: Comparison of detection powers of common evaluation methods for spray-dried and hot-melt extruded formulations. Journal of Pharmaceutical Sciences. 114 [1] (2025) 145-156 10.1016/j.xphs.2024.06.020 Open Access | |
| Minh-Dat Quoc Tang, Nhi Bao Tran, Thu-Ha Thi Nguyen, Khanh-Uyen Hoang Nguyen, Nhu-Thuy Trinh, Toi Van Vo, Makoto Kobayashi, Toru Yoshitomi, Yukio Nagasaki, Long Binh Vong. Development of oral pH-sensitive redox nanotherapeutics for gastric ulcer therapy. Journal of Controlled Release. 375 (2024) 758-766 10.1016/j.jconrel.2024.09.039 Open Access | |